SID103904592
Ligand Summary
Target Activities
MAPK8
Mitogen-activated protein kinase 8
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.6 | None, None:None:None | ||||
RPS6KA3
Ribosomal protein S6 kinase alpha-3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
CDK1
Cyclin-dependent kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
CDK2
Cyclin-dependent kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
FYN
Tyrosine-protein kinase Fyn
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
FLT1
Vascular endothelial growth factor receptor 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
FLT4
Vascular endothelial growth factor receptor 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
FLT3
Receptor-type tyrosine-protein kinase FLT3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
JAK3
Tyrosine-protein kinase JAK3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
SYK
Tyrosine-protein kinase SYK
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
JAK2
Tyrosine-protein kinase JAK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.1 | None, None:None:None | ||||
IRAK1
Interleukin-1 receptor-associated kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
TYK2
Non-receptor tyrosine-protein kinase TYK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
CSNK2A1
Casein kinase II subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
FER
Tyrosine-protein kinase Fer
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
MAPK9
Mitogen-activated protein kinase 9
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
SLK
STE20-like serine/threonine-protein kinase
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
FRK
Tyrosine-protein kinase FRK
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
CLK2
Dual specificity protein kinase CLK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
PAK4
Serine/threonine-protein kinase PAK 4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
AXL
Tyrosine-protein kinase receptor UFO
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
TAOK1
Serine/threonine-protein kinase TAO1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
PTK2B
Protein-tyrosine kinase 2-beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
NTRK3
NT-3 growth factor receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
PRKAA1
5'-AMP-activated protein kinase catalytic subunit alpha-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
AURKB
Aurora kinase B
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
AURKA
Aurora kinase A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.8 | None, None:None:None | ||||
RET
Proto-oncogene tyrosine-protein kinase receptor Ret
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.9 | None, None:None:None | ||||
ITK
Tyrosine-protein kinase ITK/TSK
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
PLK4
Serine/threonine-protein kinase PLK4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
CDK5
Cyclin-dependent-like kinase 5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
NEK4
Serine/threonine-protein kinase Nek4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||