4'-Hydroxynorendoxifen
Ligand Summary
Name: 4'-Hydroxynorendoxifen
PubChem: 73386689
ChEMBL: CHEMBL3422028
LyCHI: SP838XYUAUN3
Target Activities
CYP3A5
Cytochrome P450 3A5
2 Activities
CYP1A2
Cytochrome P450 1A2
2 Activities
CYP19A1
Aromatase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.35 | J. Med. Chem., (2015) 58:6:2623 | ||||
ESR2
Estrogen receptor beta
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 8.02 | J. Med. Chem., (2015) 58:6:2623 | ||||
ESR1
Estrogen receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 7.82 | J. Med. Chem., (2015) 58:6:2623 | ||||
CYP2A6
Cytochrome P450 2A6
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6.15 | J. Med. Chem., (2015) 58:6:2623 | ||||
CYP2D6
Cytochrome P450 2D6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6.37 | J. Med. Chem., (2015) 58:6:2623 | ||||