CHEMBL2151321
Ligand Summary
Name: CHEMBL2151321::US8486966, 1
PubChem: 59627005
Guide to Pharmacology: 8138
ChEMBL: CHEMBL2151321
LyCHI: S5YXAA3P4ULD
Target Activities
NTRK1
High affinity nerve growth factor receptor
3 Activities
ABL1
Tyrosine-protein kinase ABL1
2 Activities
BTK
Tyrosine-protein kinase BTK
2 Activities
FGR
Tyrosine-protein kinase Fgr
2 Activities
FGFR1
Fibroblast growth factor receptor 1
2 Activities
FLT3
Receptor-type tyrosine-protein kinase FLT3
2 Activities
PHKG2
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform
2 Activities
SIK1
Serine/threonine-protein kinase SIK1
2 Activities
TSSK2
Testis-specific serine/threonine-protein kinase 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.51 | |||||
WNK3
Serine/threonine-protein kinase WNK3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7 | |||||
SRC
Proto-oncogene tyrosine-protein kinase Src
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.74 | ACS Med. Chem. Lett., (2012) 3:9:705 | ||||
PTK2
Focal adhesion kinase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.76 | ACS Med. Chem. Lett., (2012) 3:9:705 | ||||
MAPK14
Mitogen-activated protein kinase 14
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.87 | ACS Med. Chem. Lett., (2012) 3:9:705 | ||||