CHEMBL4248386
Ligand Summary
Name: 2,3-dimethyl-4-(2-methyl-3-(vinylsulfonamido)phenyl)-1H-indole-7-carboxamide
PubChem: 121294143
ChEMBL: CHEMBL4248386
LyCHI: RRF7YSVWANJB
Target Activities
BTK
Tyrosine-protein kinase BTK
2 Activities
JAK3
Tyrosine-protein kinase JAK3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.96 | Bioorg Med Chem Lett, (2018) 28:18:3080 | ||||
BMX
Cytoplasmic tyrosine-protein kinase BMX
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.48 | Bioorg Med Chem Lett, (2018) 28:18:3080 | ||||
TEC
Tyrosine-protein kinase Tec
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9.05 | Bioorg Med Chem Lett, (2018) 28:18:3080 | ||||
TXK
Tyrosine-protein kinase TXK
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.64 | Bioorg Med Chem Lett, (2018) 28:18:3080 | ||||
ITK
Tyrosine-protein kinase ITK/TSK
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.08 | Bioorg Med Chem Lett, (2018) 28:18:3080 | ||||
ERBB4
Receptor tyrosine-protein kinase erbB-4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8 | Bioorg Med Chem Lett, (2018) 28:18:3080 | ||||