BAY 61-3606
Ligand Summary
Name: BAY 61-3606
PubChem: 10200390
PubChem: 52949496
PubChem: 11784504
Guide to Pharmacology: 9693
ChEMBL: CHEMBL1242100
ChEMBL: CHEMBL1190711
ChEMBL: CHEMBL541400
LyCHI: RPDMYVRX8AFU
Target Activities
SYK
Tyrosine-protein kinase SYK
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.59 | |||||
Ki | 8.12 | Chem. Biol., (2005) 12:6:621 | ||||
Ki | 8.12 | J. Med. Chem., (2012) 55:8:3614 | ||||
IC50 | 8 | Proc. Natl. Acad. Sci. U.S.A., (2007) 104:51:20523 | ||||
EC50 | 7.92 | J. Med. Chem., (2012) 55:8:3614 | ||||
MAP4K2
Mitogen-activated protein kinase kinase kinase kinase 2
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.95 | |||||
Ki | 7.8 | None, None:None:None | ||||
CHUK
Inhibitor of nuclear factor kappa-B kinase subunit alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.35 | |||||
CLK4
Dual specificity protein kinase CLK4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8 | None, None:None:None | ||||
GSK3B
Glycogen synthase kinase-3 beta
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
CDC7
Cell division cycle 7-related protein kinase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
NEK4
Serine/threonine-protein kinase Nek4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||