CHEMBL2418806
Ligand Summary
Name: N-(4-Methylphenyl)-4-[(2,3-dimethyl-1-piperidinyl)carbonyl]-1,3-thiazol-2-amine
PubChem: 71818431
ChEMBL: CHEMBL2418806
LyCHI: RN98RGR781WB
Target Activities
CACNA1C
Voltage-dependent L-type calcium channel subunit alpha-1C
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5 | Bioorg. Med. Chem. Lett., (2013) 23:17:4979 | ||||
TRPV1
Transient receptor potential cation channel subfamily V member 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5.9 | Bioorg. Med. Chem. Lett., (2013) 23:17:4979 | ||||
TRPA1
Transient receptor potential cation channel subfamily A member 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5.1 | Bioorg. Med. Chem. Lett., (2013) 23:17:4979 | ||||
TRPV4
Transient receptor potential cation channel subfamily V member 4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5.2 | Bioorg. Med. Chem. Lett., (2013) 23:17:4979 | ||||
TRPC6
Short transient receptor potential channel 6
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.1 | Bioorg. Med. Chem. Lett., (2013) 23:17:4979 | ||||
TRPC3
Short transient receptor potential channel 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.6 | Bioorg. Med. Chem. Lett., (2013) 23:17:4979 | ||||