phorbol 12-myristate 13-acetate
Ligand Summary
Name: phorbol 12-myristate 13-acetate
PubChem: 27924
Guide to Pharmacology: 2341
ChEMBL: CHEMBL279115
LyCHI: RKDKAMM28NUC
Target Activities
TRPV4
Transient receptor potential cation channel subfamily V member 4
2 Activities
PRKCA
Protein kinase C alpha type
2 Activities
KCNT2
Potassium channel subfamily T member 2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
7.92 | ||||||
PRKCG
Protein kinase C gamma type
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.31 | Bioorg. Med. Chem. Lett., (2001) 11:8:955 | ||||
PRKCD
Protein kinase C delta type
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 9.1 | Bioorg. Med. Chem. Lett., (2001) 11:8:955 | ||||
PRKCB
Protein kinase C beta type
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.74 | Bioorg. Med. Chem. Lett., (2001) 11:8:955 | ||||
PRKCE
Protein kinase C epsilon type
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 9.35 | Bioorg. Med. Chem. Lett., (2001) 11:8:955 | ||||
RASGRP3
Ras guanyl-releasing protein 3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 7.09 | J Med Chem, (2018) 61:14:6261 | ||||