Pharos : Ligand Details - RHDD5N5DSTYC

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: UNC0638

PubChem: 46224516

Guide to Pharmacology: 7015

ChEMBL: CHEMBL1231795

LyCHI: RHDD5N5DSTYC

Target Activities

Explore Associated and Predicted Targets

EHMT2

Tchem

Histone-lysine N-methyltransferase EHMT2

24 Activities

Items per page:

1 – 10 of 24

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.82			21743462

Ki	8.52			21743462

IC50	8.6		MedChemComm, (2014) 5:12:1821	25750706

Ki	8.43		Eur. J. Med. Chem., (2012) 56:None:179	22975593

Ki	8.43		Bioorg Med Chem, (2016) 24:22:6102	27720557

IC50	7.92		J. Med. Chem., (2011) 54:17:6139	21780790

IC50	7.82		Eur J Med Chem, (2019) 179:None:537	31276898

IC50	7.82		J Med Chem, (2019) 62:5:2666	30753076

IC50	7.6		J Med Chem, (2019) 62:5:2666	30753076

IC50	7.58		Bioorg Med Chem Lett, (2019) 29:17:2516	31350126

EHMT1

Tchem

Histone-lysine N-methyltransferase EHMT1

6 Activities

Items per page:

1 – 6 of 6

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.72			21743462

IC50	7.89		Bioorg Med Chem Lett, (2019) 29:17:2516	31350126

IC50	7.72		Eur. J. Med. Chem., (2012) 56:None:179	22975593

IC50	7.72		MedChemComm, (2012) 3:2:135

IC50	7.72		Bioorg Med Chem, (2017) 25:17:4579	28739157

IC50	7.72		J Med Chem, (2019) 62:5:2666	30753076