Pharos : Ligand Details - RHDD5N5DSTYC

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Ligand Summary

Ligand Structure

chemical structure image

Synonyms & Links

Name: UNC0638

PubChem: 46224516

Guide to Pharmacology: 7015

ChEMBL: CHEMBL1231795

LyCHI: RHDD5N5DSTYC

Target Activities

EHMT2

Tchem

Histone-lysine N-methyltransferase EHMT2

17 Activities

Items per page:

1 – 10 of 17

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.21		Bioorg Med Chem, (2016) 24:22:6102	27720557

IC50	6.62		J. Med. Chem., (2011) 54:17:6139	21780790

IC50	6.68		J. Med. Chem., (2011) 54:17:6139	21780790

IC50	6.92		J. Med. Chem., (2011) 54:17:6139	21780790

IC50	7.09		J. Med. Chem., (2011) 54:17:6139	21780790

IC50	7.09		Eur. J. Med. Chem., (2012) 56:None:179	22975593

IC50	7.09		Eur. J. Med. Chem., (2012) 56:None:179	22975593

IC50	7.09		J. Med. Chem., (2013) 56:21:8931	24102134

IC50	7.16		J. Med. Chem., (2011) 54:17:6139	21780790

IC50	7.23		J. Med. Chem., (2011) 54:17:6139	21780790

EHMT1

Tchem

Histone-lysine N-methyltransferase EHMT1

3 Activities

Items per page:

1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.72		MedChemComm, (2012) 3:2:135

IC50	7.72		Eur. J. Med. Chem., (2012) 56:None:179	22975593

IC50	7.71999979			21743462