UNC0638
Ligand Summary
Name: UNC0638
PubChem: 46224516
Guide to Pharmacology: 7015
ChEMBL: CHEMBL1231795
LyCHI: RHDD5N5DSTYC
Target Activities
EHMT2
Histone-lysine N-methyltransferase EHMT2
24 Activities
Items per page:
1 – 10 of 24
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.82 | |||||
Ki | 8.52 | |||||
IC50 | 8.6 | MedChemComm, (2014) 5:12:1821 | ||||
Ki | 8.43 | Eur. J. Med. Chem., (2012) 56:None:179 | ||||
Ki | 8.43 | Bioorg Med Chem, (2016) 24:22:6102 | ||||
IC50 | 7.92 | J. Med. Chem., (2011) 54:17:6139 | ||||
IC50 | 7.82 | Eur J Med Chem, (2019) 179:None:537 | ||||
IC50 | 7.82 | J Med Chem, (2019) 62:5:2666 | ||||
IC50 | 7.6 | J Med Chem, (2019) 62:5:2666 | ||||
IC50 | 7.58 | Bioorg Med Chem Lett, (2019) 29:17:2516 | ||||
EHMT1
Histone-lysine N-methyltransferase EHMT1
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.72 | |||||
IC50 | 7.89 | Bioorg Med Chem Lett, (2019) 29:17:2516 | ||||
IC50 | 7.72 | Eur. J. Med. Chem., (2012) 56:None:179 | ||||
IC50 | 7.72 | MedChemComm, (2012) 3:2:135 | ||||
IC50 | 7.72 | Bioorg Med Chem, (2017) 25:17:4579 | ||||
IC50 | 7.72 | J Med Chem, (2019) 62:5:2666 | ||||