(E)-Norendoxifen
Ligand Summary
Target Activities
CYP19A1
Aromatase
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.32 | J. Med. Chem., (2013) 56:11:4611 | ||||
IC50 | 7.12 | J. Med. Chem., (2013) 56:11:4611 | ||||
IC50 | 7.12 | Bioorg Med Chem, (2016) 24:21:5400 | ||||
IC50 | 7.05 | J. Med. Chem., (2013) 56:11:4611 | ||||
IC50 | 6.99 | J. Med. Chem., (2015) 58:6:2623 | ||||