Pharos : Ligand Details - QW52DF1DQMCJ

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Ligand Summary

Ligand Structure

chemical structure image

Synonyms & Links

Name: 8-Cyclohexylmethyl-2-(2-fluoro-phenyl)-6,7,8,9-tetrahydro-5H-1,3a,5,8-tetraaza-cyclopenta[a]naphthalen-4-one

PubChem: 11047145

PubChem: 11783674

ChEMBL: CHEMBL146230

ChEMBL: CHEMBL356161

LyCHI: QW52DF1DQMCJ

Target Activities

GABRA2

Tclin

Gamma-aminobutyric acid receptor subunit alpha-2

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	6.7		J. Med. Chem., (2002) 45:23:5043	12408715

EC50	7.7		J. Med. Chem., (2002) 45:23:5043	12408715

GABRA3

Tclin

Gamma-aminobutyric acid receptor subunit alpha-3

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	6.67		J. Med. Chem., (2002) 45:23:5043	12408715

EC50	7.7		J. Med. Chem., (2002) 45:23:5043	12408715

GABRA5

Tclin

Gamma-aminobutyric acid receptor subunit alpha-5

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	6.64		J. Med. Chem., (2002) 45:23:5043	12408715

EC50	7.13		J. Med. Chem., (2002) 45:23:5043	12408715

GABRA1

Tclin

Gamma-aminobutyric acid receptor subunit alpha-1

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	6.9		J. Med. Chem., (2002) 45:23:5043	12408715

EC50	7.75		J. Med. Chem., (2002) 45:23:5043	12408715