CHEMBL4078014
Ligand Summary
Name: 3-(4-((4-(2-fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)methyl)benzoyl)piperazin-1-yl)methyl)phenyl)-N-hydroxyacrylamide
PubChem: 132576507
ChEMBL: CHEMBL4078014
LyCHI: QVLHFMVF5WCT
Target Activities
PARP2
Poly [ADP-ribose] polymerase 2
2 Activities
HDAC1
Histone deacetylase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.42 | Bioorg Med Chem, (2017) 25:15:4100 | ||||
HDAC6
Histone deacetylase 6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.99 | Bioorg Med Chem, (2017) 25:15:4100 | ||||
PARP1
Poly [ADP-ribose] polymerase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.82 | Bioorg Med Chem, (2017) 25:15:4100 | ||||