CHEMBL3289421
Ligand Summary
Name: 12-Oxo-N-(2-pyrrolidin-1-ylethyl)-12H-benzo[g]pyrido[2,1-b]-quinazoline-4-carboxamide
PubChem: 90644357
ChEMBL: CHEMBL3289421
LyCHI: QSUARS2R8KSG
Target Activities
POLR1A
DNA-directed RNA polymerase I subunit RPA1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.05 | J. Med. Chem., (2014) 57:11:4950 | ||||