Pharos : Ligand Details

Target Activities

Explore Associated and Predicted Targets

PRKCQ

Tchem

Protein kinase C theta type

6 Activities

Items per page:

1 – 6 of 6

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	9		19827831

Ki	9.2	None, None:None:None

IC50	9	J. Med. Chem., (2009) 52:20:6193	19827831

IC50	9	J. Med. Chem., (2011) 54:17:6028	21797275

IC50	9	Bioorg Med Chem Lett, (2017) 27:4:781	28131714

Kd	7.89	Science, (2017) 358:6367:None	29191878

PRKCA

Tchem

Protein kinase C alpha type

5 Activities

Items per page:

1 – 5 of 5

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	8.68		19827831

IC50	8.68	J. Med. Chem., (2009) 52:20:6193	19827831

IC50	8.68	J. Med. Chem., (2011) 54:17:6028	21797275

IC50	8.68	Bioorg Med Chem Lett, (2017) 27:4:781	28131714

Kd	7.89	Science, (2017) 358:6367:None	29191878

PRKCB

Tchem

Protein kinase C beta type

5 Activities

Items per page:

1 – 5 of 5

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	8.7		19827831

IC50	8.7	J. Med. Chem., (2009) 52:20:6193	19827831

IC50	8.7	J. Med. Chem., (2011) 54:17:6028	21797275

IC50	8.7	Bioorg Med Chem Lett, (2017) 27:4:781	28131714

Kd	7.62	Science, (2017) 358:6367:None	29191878

PRKCD

Tclin

Protein kinase C delta type

5 Activities

Items per page:

1 – 5 of 5

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	8.89		19827831

IC50	8.89	J. Med. Chem., (2009) 52:20:6193	19827831

IC50	8.89	J. Med. Chem., (2011) 54:17:6028	21797275

IC50	8.89	Bioorg Med Chem Lett, (2017) 27:4:781	28131714

Kd	8.3	Science, (2017) 358:6367:None	29191878

PRKCE

Tchem

Protein kinase C epsilon type

4 Activities

Items per page:

1 – 4 of 4

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	8.21		19827831

IC50	8.21	J. Med. Chem., (2009) 52:20:6193	19827831

IC50	8.21	J. Med. Chem., (2011) 54:17:6028	21797275

IC50	8.21	Bioorg Med Chem Lett, (2017) 27:4:781	28131714

PRKCH

Tchem

Protein kinase C eta type

4 Activities

Items per page:

1 – 4 of 4

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	8.21		19827831

IC50	8.21	J. Med. Chem., (2009) 52:20:6193	19827831

IC50	8.21	J. Med. Chem., (2011) 54:17:6028	21797275

IC50	8.21	Bioorg Med Chem Lett, (2017) 27:4:781	28131714

PRKCG

Tchem

Protein kinase C gamma type

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.9		None, None:None:None

PIM2

Tchem

Serine/threonine-protein kinase pim-2

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	8.8		None, None:None:None

MINK1

Tchem

Misshapen-like kinase 1

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	8.1		None, None:None:None