CHEMBL4648912
Ligand Summary
Name: N-(1-(1,1-Di(pyridin-2-yl)ethyl)-6-(1-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-3-yl)-1H-indol-4-yl)-ethanesulfonamide
PubChem: 146036007
ChEMBL: CHEMBL4648912
LyCHI: QC1M8HCPY8F3
Target Activities
BRD4
Bromodomain-containing protein 4
2 Activities
EP300
Histone acetyltransferase p300
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.43 | J Med Chem, (2020) 63:13:7186 | ||||
TAF1
Transcription initiation factor TFIID subunit 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.04 | J Med Chem, (2020) 63:13:7186 | ||||