Pharos : Ligand Details - QAJV4C8T6J25

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: UNC1999

PubChem: 72551585

Guide to Pharmacology: 8237

ChEMBL: CHEMBL3414619

LyCHI: QAJV4C8T6J25

Target Activities

Explore Associated and Predicted Targets

EZH2

Tclin

Histone-lysine N-methyltransferase EZH2

3 Activities

Items per page:

1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.7			23614352

Ki	8.34		J. Med. Chem., (2015) 58:4:1596	25406853

IC50	6.91		J. Med. Chem., (2015) 58:4:1596	25406853

EZH1

Tchem

Histone-lysine N-methyltransferase EZH1

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.16		J Med Chem, (2016) 59:16:7617	27468126