tomivosertib
Ligand Summary
Name: tomivosertib
PubChem: 118598754
PubChem: 118598855
Guide to Pharmacology: 10167
ChEMBL: CHEMBL4073443
ChEMBL: CHEMBL4298140
LyCHI: Q8GZR1M2KVNX
Target Activities
MKNK1
MAP kinase-interacting serine/threonine-protein kinase 1
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.62 | |||||
IC50 | 8.7 | Eur J Med Chem, (2019) 163:None:413 | ||||
IC50 | 8.62 | J Med Chem, (2018) 61:8:3516 | ||||
Ki | 8.3 | Bioorg Med Chem Lett, (2019) 29:18:2650 | ||||
MKNK2
MAP kinase-interacting serine/threonine-protein kinase 2
4 Activities
CLK4
Dual specificity protein kinase CLK4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.1 | |||||
STK17A
Serine/threonine-protein kinase 17A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.89 | |||||