SID103904605
Ligand Summary
Target Activities
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
RPS6KA3
Ribosomal protein S6 kinase alpha-3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9 | None, None:None:None | ||||
CDK2
Cyclin-dependent kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.8 | None, None:None:None | ||||
DAPK3
Death-associated protein kinase 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.9 | None, None:None:None | ||||
JAK3
Tyrosine-protein kinase JAK3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
SYK
Tyrosine-protein kinase SYK
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
GSK3A
Glycogen synthase kinase-3 alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.9 | None, None:None:None | ||||
JAK2
Tyrosine-protein kinase JAK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
CDK7
Cyclin-dependent kinase 7
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
PRKACA
cAMP-dependent protein kinase catalytic subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
CLK2
Dual specificity protein kinase CLK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
PAK4
Serine/threonine-protein kinase PAK 4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
STK17A
Serine/threonine-protein kinase 17A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
MELK
Maternal embryonic leucine zipper kinase
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.8 | None, None:None:None | ||||
GSK3B
Glycogen synthase kinase-3 beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
MAP4K5
Mitogen-activated protein kinase kinase kinase kinase 5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
MAP4K2
Mitogen-activated protein kinase kinase kinase kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.7 | None, None:None:None | ||||
MINK1
Misshapen-like kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
STK3
Serine/threonine-protein kinase 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
CDK9
Cyclin-dependent kinase 9
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.7 | None, None:None:None | ||||
CDC7
Cell division cycle 7-related protein kinase
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.6 | None, None:None:None | ||||
PRKD3
Serine/threonine-protein kinase D3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
ROCK2
Rho-associated protein kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
PRKX
cAMP-dependent protein kinase catalytic subunit PRKX
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||