Pharos : Ligand Details - P8PWSR24G7GT

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: (S)-3-(1H-Indol-3-yl)-2-[(R)-3-mercapto-2-((S)-5-methoxy-indan-1-yl)-propionylamino]-propionic acid

PubChem: 44303110

ChEMBL: CHEMBL305388

LyCHI: P8PWSR24G7GT

Target Activities

Explore Associated and Predicted Targets

ECE1

Tchem

Endothelin-converting enzyme 1

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	8		J. Med. Chem., (2005) 48:21:6523	16220969

Ki	6.75		Bioorg. Med. Chem. Lett., (2002) 12:15:2001	12113828

ACE

Tclin

Angiotensin-converting enzyme

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	8.89		J. Med. Chem., (2005) 48:21:6523	16220969

MME

Tclin

Neprilysin

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.62		J. Med. Chem., (2005) 48:21:6523	16220969