GW9508
Ligand Summary
Name: GW9508
PubChem: 11595431
Guide to Pharmacology: 1050
ChEMBL: CHEMBL207881
LyCHI: N7SA8ZVAG8UY
Target Activities
FFAR1
Free fatty acid receptor 1
13 Activities
Items per page:
1 – 10 of 13
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
- | 7.3 | |||||
EC50 | 7.89 | Bioorg. Med. Chem. Lett., (2014) 24:13:2949 | ||||
EC50 | 7.55 | J. Med. Chem., (2012) 55:9:4511 | ||||
EC50 | 7.55 | J. Med. Chem., (2016) 59:10:4849 | ||||
EC50 | 7.54 | ACS Med. Chem. Lett., (2010) 1:7:345 | ||||
EC50 | 7.32 | J. Med. Chem., (2008) 51:22:7061 | ||||
EC50 | 7.32 | J. Med. Chem., (2011) 54:19:6691 | ||||
EC50 | 7.32 | Bioorg Med Chem Lett, (2018) 28:15:2599 | ||||
EC50 | 7.3 | ACS Med Chem Lett, (2017) 8:12:1336 | ||||
EC50 | 7.19 | Bioorg. Med. Chem. Lett., (2006) 16:7:1840 | ||||