CHEMBL4450921
Ligand Summary
Name: 3-(7-Methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-(((R)-4-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b]-[1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoic Acid
PubChem: 118170387
ChEMBL: CHEMBL4450921
LyCHI: MNQSKVQULJFB
Target Activities
NFE2L2
Nuclear factor erythroid 2-related factor 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
EC50 | 7.96 | J Med Chem, (2019) 62:9:4683 | ||||
KEAP1
Kelch-like ECH-associated protein 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8 | J Med Chem, (2019) 62:9:4683 | ||||