L-796449
Ligand Summary
Name: L-796449
PubChem: 9891946
Guide to Pharmacology: 2689
ChEMBL: CHEMBL278994
LyCHI: MLJBWZZWNBJ9
Target Activities
PPARD
Peroxisome proliferator-activated receptor delta
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
8.7 | ||||||
EC50 | 8.22 | Bioorg. Med. Chem. Lett., (2003) 13:7:1277 | ||||
IC50 | 8.22 | Bioorg. Med. Chem. Lett., (2003) 13:7:1277 | ||||
IC50 | 8.22 | Bioorg. Med. Chem., (2012) 20:11:3523 | ||||
EC50 | 8.1 | J. Med. Chem., (2000) 43:4:527 | ||||
EC50 | 8.1 | Eur. J. Med. Chem., (2012) 53:None:190 | ||||
PPARG
Peroxisome proliferator-activated receptor gamma
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
8.7 | ||||||
EC50 | 8.28 | J. Med. Chem., (2000) 43:4:527 | ||||
EC50 | 8.05 | Bioorg. Med. Chem. Lett., (2003) 13:7:1277 | ||||
IC50 | 7.03 | Bioorg. Med. Chem. Lett., (2003) 13:7:1277 | ||||
IC50 | 7.03 | Eur. J. Med. Chem., (2011) 46:6:2513 | ||||
IC50 | 7.03 | Bioorg. Med. Chem., (2012) 20:11:3523 | ||||
PPARA
Peroxisome proliferator-activated receptor alpha
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
EC50 | 8.39 | J. Med. Chem., (2000) 43:4:527 | ||||
EC50 | 7.75 | Bioorg. Med. Chem. Lett., (2003) 13:7:1277 | ||||
IC50 | 7.27 | Bioorg. Med. Chem. Lett., (2003) 13:7:1277 | ||||
IC50 | 7.27 | Bioorg. Med. Chem., (2012) 20:11:3523 | ||||