CHEMBL4215326
Ligand Summary
Name: 6-Methoxy-7-[(2-methyl-2-azaspiro[3.3]heptan-6-yl)oxy]-2-(5-methyl-2-furyl)-N-(1-methyl-4-piperidyl)quinolin-4-amine
PubChem: 129072680
ChEMBL: CHEMBL4215326
LyCHI: MJGFTC6HH632
Target Activities
DNMT1
DNA (cytosine-5)-methyltransferase 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.68 | J Med Chem, (2018) 61:15:6546 | ||||
EHMT2
Histone-lysine N-methyltransferase EHMT2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.46 | J Med Chem, (2018) 61:15:6546 | ||||