CHEMBL4099681
Ligand Summary
Name: 4-(5-(2,6-Difluoro-3-hydroxybenzoyl)thiophen-2-yl)-2,3-difluorophenyl sulfamate
PubChem: 137661419
ChEMBL: CHEMBL4099681
LyCHI: MAU8FD5VCRWT
Target Activities
HSD17B1
Estradiol 17-beta-dehydrogenase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.57 | J Med Chem, (2017) 60:9:4086 | ||||
HSD17B2
Estradiol 17-beta-dehydrogenase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.63 | J Med Chem, (2017) 60:9:4086 | ||||
STS
Steryl-sulfatase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.98 | J Med Chem, (2017) 60:9:4086 | ||||