CHEMBL247920
Ligand Summary
Name: 2-[3-[2-(5-ethyl-3,4-diphenylpyrazol-1-yl)phenyl]phenoxy]acetic acid
PubChem: 16122583
ChEMBL: CHEMBL247920
LyCHI: M9G6WXGT96UW
Target Activities
FABP4
Fatty acid-binding protein, adipocyte
7 Activities
Items per page:
1 – 7 of 7
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.13 | Bioorg. Med. Chem. Lett., (2007) 17:12:3511 | ||||
Ki | 7.82 | Bioorg. Med. Chem. Lett., (2011) 21:10:2949 | ||||
Ki | 6.8 | ACS Med. Chem. Lett., (2016) 7:4:435 | ||||
IC50 | 6.66 | Bioorg. Med. Chem. Lett., (2013) 23:6:1662 | ||||
Ki | 6.66 | Bioorg. Med. Chem., (2016) 24:18:4310 | ||||
Ki | 6.6 | J Med Chem, (2020) 63:8:4090 | ||||
Kd | 6.6 | J Med Chem, (2020) 63:8:4090 | ||||
FABP3
Fatty acid-binding protein, heart
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6.6 | Bioorg. Med. Chem. Lett., (2007) 17:12:3511 | ||||
FABP5
Fatty acid-binding protein 5
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6.46 | Bioorg. Med. Chem. Lett., (2007) 17:12:3511 | ||||