adavosertib
Ligand Summary
Name: adavosertib
PubChem: 24856436
Guide to Pharmacology: 7702
ChEMBL: CHEMBL1976040
LyCHI: LXRDJN426DS6
Target Activities
WEE1
Wee1-like protein kinase
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.29 | |||||
Kd | 8.49 | J Med Chem, (2017) 60:18:7863 | ||||
IC50 | 8.28 | Bioorg Med Chem, (2018) 26:14:4014 | ||||
Kd | 7.92 | Science, (2017) 358:6367:None | ||||
Kd | 7.87 | J Med Chem, (2017) 60:18:7863 | ||||
WEE2
Wee1-like protein kinase 2
2 Activities
JAK3
Tyrosine-protein kinase JAK3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.58 | J Med Chem, (2017) 60:18:7863 | ||||
PLK1
Serine/threonine-protein kinase PLK1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.52 | J Med Chem, (2017) 60:18:7863 | ||||
ADK
Adenosine kinase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.89 | Science, (2017) 358:6367:None | ||||