CHEMBL2017835
Ligand Summary
Name: (4S)-6-{2-[(2R)-2-(3,5-dimethylbenzyl)piperidin-1-yl]-2-oxoethyl}-4-(1H-indazol-3-ylmethyl)-1-phenyl-4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5(6H)-one
PubChem: 46235271
ChEMBL: CHEMBL2017835
LyCHI: LWGMAB1CHUQK
Target Activities
CCKAR
Cholecystokinin receptor type A
18 Activities
Items per page:
1 – 10 of 18
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.15 | J. Med. Chem., (2015) 58:24:9562 | ||||
EC50 | 7.16 | J. Med. Chem., (2015) 58:24:9562 | ||||
IC50 | 7.21 | J. Med. Chem., (2015) 58:24:9562 | ||||
IC50 | 7.37 | J. Med. Chem., (2015) 58:24:9562 | ||||
IC50 | 7.46 | J. Med. Chem., (2015) 58:24:9562 | ||||
Ki | 7.54 | J. Med. Chem., (2015) 58:24:9562 | ||||
IC50 | 7.56 | J. Med. Chem., (2015) 58:24:9562 | ||||
IC50 | 7.69 | Bioorg. Med. Chem. Lett., (2012) 22:8:2943 | ||||
IC50 | 8 | J. Med. Chem., (2015) 58:24:9562 | ||||
IC50 | 8.14 | J. Med. Chem., (2015) 58:24:9562 | ||||