CHEMBL4277352
Ligand Summary
Name: N2,N4-bis(3,3-difluorocyclopentyl)-6-[6-(trifluoromethyl)-2-pyridyl]-1,3,5-triazine-2,4-diamine
PubChem: 86580656
ChEMBL: CHEMBL4277352
LyCHI: LLLH2NF8NZXN
Target Activities
IDH1
Isocitrate dehydrogenase [NADP] cytoplasmic
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | ACS Med Chem Lett, (2020) 11:2:101 | ||||
IDH2
Isocitrate dehydrogenase [NADP], mitochondrial
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.05 | ACS Med Chem Lett, (2020) 11:2:101 | ||||