guggulsterone
Ligand Summary
Name: guggulsterone
PubChem: 6439929
Guide to Pharmacology: 2745
ChEMBL: CHEMBL402063
LyCHI: L818G9DRGCV3
Target Activities
NR1H4
Bile acid receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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- | 5 | |||||
NR3C2
Mineralocorticoid receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.41 | J. Med. Chem., (2005) 48:22:6948 | ||||
NR1I2
Nuclear receptor subfamily 1 group I member 2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 8.62 | J. Med. Chem., (2005) 48:22:6948 | ||||