CHEMBL1945803
Ligand Summary
Name: 9-Chloro-2-({5-[3-(dimethylamino)propyl]pyridin-3-yl}-amino)-5,7-dihydro-6H-pyrimido[5,4-d][1]benzazepine-6-thione
PubChem: 46235770
ChEMBL: CHEMBL1945803
LyCHI: L6ADBJG8NHSZ
Target Activities
PDGFRB
Platelet-derived growth factor receptor beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.57 | J. Med. Chem., (2012) 55:1:197 | ||||
KIT
Mast/stem cell growth factor receptor Kit
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.7 | J. Med. Chem., (2012) 55:1:197 | ||||
KDR
Vascular endothelial growth factor receptor 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.96 | J. Med. Chem., (2012) 55:1:197 | ||||
PLK1
Serine/threonine-protein kinase PLK1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 9 | J. Med. Chem., (2012) 55:1:197 | ||||
FGFR1
Fibroblast growth factor receptor 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.96 | J. Med. Chem., (2012) 55:1:197 | ||||