CHEMBL445691
Ligand Summary
Name: (R)-methyl 4-(2-(3-(2-fluoro-6-(trifluoromethyl)benzyl)-5-(2-chlorophenyl)-2,6-dioxo-2,3-dihydropyrimidin-1(6H)-yl)-1-phenylethylamino)butanoate
PubChem: 44576678
ChEMBL: CHEMBL445691
LyCHI: L3ACBT8LA688
Target Activities
CYP3A4
Cytochrome P450 3A4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.89 | Bioorg. Med. Chem. Lett., (2008) 18:11:3301 | ||||
GNRHR
Gonadotropin-releasing hormone receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.18 | Bioorg. Med. Chem. Lett., (2008) 18:11:3301 | ||||