CHEMBL464552
Ligand Summary
Name: GSK-1838705A
PubChem: 25182616
Guide to Pharmacology: 5683
ChEMBL: CHEMBL464552
LyCHI: KNPYT7U7AQ2J
Target Activities
IGF1R
Insulin-like growth factor 1 receptor
4 Activities
INSR
Insulin receptor
3 Activities
ALK
ALK tyrosine kinase receptor
2 Activities
INSRR
Insulin receptor-related protein
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.07 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
MYLK
Myosin light chain kinase, smooth muscle
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.96 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
ROS1
Proto-oncogene tyrosine-protein kinase ROS
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.82 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
LTK
Leukocyte tyrosine kinase receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.96 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CLK1
Dual specificity protein kinase CLK1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.68 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
FER
Tyrosine-protein kinase Fer
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.03 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CLK2
Dual specificity protein kinase CLK2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.8 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
RPS6KA1
Ribosomal protein S6 kinase alpha-1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 5.80000019 | |||||