SU6656
Ligand Summary
Name: SU6656
PubChem: 5312137
Guide to Pharmacology: 6044
ChEMBL: CHEMBL605003
LyCHI: KHM7MCDX48PH
Target Activities
AURKB
Aurora kinase B
2 Activities
AURKC
Aurora kinase C
2 Activities
YES1
Tyrosine-protein kinase Yes
2 Activities
BRSK2
Serine/threonine-protein kinase BRSK2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7 | |||||
LCK
Tyrosine-protein kinase Lck
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.82 | |||||
LYN
Tyrosine-protein kinase Lyn
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.89 | |||||
SRC
Proto-oncogene tyrosine-protein kinase Src
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.14 | |||||
CYP1A2
Cytochrome P450 1A2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 6.5 | None, None:None:None | ||||