CHEMBL380192
Ligand Summary
Name: 7-(3-hydroxypropylthio)-4-isobutyl-2-methyl-6-(naphthalen-1-ylmethyl)-2H-pyrrolo[3,4-d]pyridazin-1(6H)-one
PubChem: 5282542
ChEMBL: CHEMBL380192
LyCHI: KH7LJSMN73BL
Target Activities
SLC16A1
Monocarboxylate transporter 1
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 10.02 | Nat. Chem. Biol., (2005) 1:7:371 | ||||
Ki | 10 | Bioorg. Med. Chem. Lett., (2006) 16:8:2260 | ||||
Ki | 9.15 | Nat. Chem. Biol., (2005) 1:7:371 | ||||
EC50 | 8.3 | MedChemComm, (2016) 7:5:900 | ||||
IC50 | 6.98 | J. Med. Chem., (2014) 57:17:7317 | ||||