K-252a
Ligand Summary
Target Activities
NTRK1
High affinity nerve growth factor receptor
3 Activities
MYLK
Myosin light chain kinase, smooth muscle
2 Activities
CDK4
Cyclin-dependent kinase 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.85 | Science, (2017) 358:6367:None | ||||
PRKAG2
5'-AMP-activated protein kinase subunit gamma-2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 6.06 | Science, (2017) 358:6367:None | ||||
AAK1
AP2-associated protein kinase 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
IRAK4
Interleukin-1 receptor-associated kinase 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.05 | Science, (2017) 358:6367:None | ||||
CLK4
Dual specificity protein kinase CLK4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.82 | Science, (2017) 358:6367:None | ||||
CLK1
Dual specificity protein kinase CLK1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8 | Science, (2017) 358:6367:None | ||||
TNIK
TRAF2 and NCK-interacting protein kinase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8 | Science, (2017) 358:6367:None | ||||
STK4
Serine/threonine-protein kinase 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.54 | Science, (2017) 358:6367:None | ||||
NEK7
Serine/threonine-protein kinase Nek7
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 8.52 | Science, (2017) 358:6367:None | ||||
MARK4
MAP/microtubule affinity-regulating kinase 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.55 | Science, (2017) 358:6367:None | ||||
MAP4K4
Mitogen-activated protein kinase kinase kinase kinase 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.72 | Science, (2017) 358:6367:None | ||||
ERN1
Serine/threonine-protein kinase/endoribonuclease IRE1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.72 | Science, (2017) 358:6367:None | ||||
AURKA
Aurora kinase A
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.7 | Science, (2017) 358:6367:None | ||||
Q6ZSR9
Uncharacterized protein FLJ45252
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 7.68 | Science, (2017) 358:6367:None | ||||