CHEMBL179503
Ligand Summary
Name: [3-(2-{5-tert-Butyl-3-[(4-methyl-furazan-3-ylmethyl)-amino]-2-oxo-2H-pyrazin-1-yl}-butyrylamino)-4-carboxy-2-oxo-butyl]-methyl-pentyl-ammonium chloride
PubChem: 11467504
ChEMBL: CHEMBL179503
LyCHI: KA2VH7AQT61S
Target Activities
CASP4
Caspase-4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9.3 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||
CASP5
Caspase-5
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9.09 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||
CASP6
Caspase-6
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.46 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||
CASP7
Caspase-7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 10.05 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||
CASP8
Caspase-8
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.39 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||
CASP1
Caspase-1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9.96 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||
CASP10
Caspase-10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.53 | Bioorg. Med. Chem. Lett., (2005) 15:4:1173 | ||||