US8937193, 6i
Ligand Summary
Target Activities
BCL2L1
Bcl-2-like protein 1
7 Activities
Items per page:
1 – 7 of 7
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.12 | J Med Chem, (2017) 60:3:821 | ||||
Ki | 7.12 | Eur J Med Chem, (2019) 177:None:63 | ||||
Ki | 6.64 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.47 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.47 | None, (2015) None:None:None | ||||
Kd | 6.35 | J. Med. Chem., (2010) 53:22:8000 | ||||
Kd | 6.35 | None, (2015) None:None:None | ||||
MCL1
Induced myeloid leukemia cell differentiation protein Mcl-1
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.6 | J Med Chem, (2017) 60:3:821 | ||||
Ki | 7.6 | Eur J Med Chem, (2019) 177:None:63 | ||||
Ki | 6.8 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.62 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.62 | None, (2015) None:None:None | ||||
BCL2
Apoptosis regulator Bcl-2
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.51 | J Med Chem, (2017) 60:3:821 | ||||
Ki | 7.51 | Eur J Med Chem, (2019) 177:None:63 | ||||
Ki | 6.72 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.54 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.54 | None, (2015) None:None:None | ||||
BCL2A1
Bcl-2-related protein A1
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.91 | J Med Chem, (2017) 60:3:821 | ||||
Ki | 6.37 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.19 | J. Med. Chem., (2010) 53:22:8000 | ||||
IC50 | 6.19 | None, (2015) None:None:None | ||||