Ergocornine
Ligand Summary
Target Activities
DRD2
D(2) dopamine receptor
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.78 | None, None:None:None | ||||
IC50 | 8.3 | None, None:None:None | ||||
HTR2B
5-hydroxytryptamine receptor 2B
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.16 | None, None:None:None | ||||
IC50 | 7.96 | None, None:None:None | ||||
DRD3
D(3) dopamine receptor
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.01 | None, None:None:None | ||||
IC50 | 8.54 | None, None:None:None | ||||
ADRA2A
Alpha-2A adrenergic receptor
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.63 | None, None:None:None | ||||
IC50 | 8.2 | None, None:None:None | ||||
ADRA1D
Alpha-1D adrenergic receptor
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.06 | None, None:None:None | ||||
IC50 | 7.75 | None, None:None:None | ||||
ADRA2B
Alpha-2B adrenergic receptor
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.86 | None, None:None:None | ||||
IC50 | 8.52 | None, None:None:None | ||||
HTR2A
5-hydroxytryptamine receptor 2A
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.1 | None, None:None:None | ||||
IC50 | 7.55 | None, None:None:None | ||||
HTR6
5-hydroxytryptamine receptor 6
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.15 | None, None:None:None | ||||
IC50 | 7.82 | None, None:None:None | ||||
ADRA2C
Alpha-2C adrenergic receptor
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.62 | None, None:None:None | ||||
IC50 | 7.77 | None, None:None:None | ||||
CYP3A4
Cytochrome P450 3A4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.3 | None, None:None:None | ||||
HTR2C
5-hydroxytryptamine receptor 2C
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.26 | None, None:None:None | ||||