BAY-299
Ligand Summary
Name: BAY-299
PubChem: 122705990
Guide to Pharmacology: 9524
ChEMBL: CHEMBL4086276
LyCHI: JHD7SC6KYURG
Target Activities
BRD1
Bromodomain-containing protein 1
13 Activities
Items per page:
1 – 10 of 13
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.22 | |||||
IC50 | 8.22 | J Med Chem, (2017) 60:1:157 | ||||
Kd | 7.44 | J Med Chem, (2017) 60:9:4002 | ||||
Kd | 7.43 | J Med Chem, (2017) 60:9:4002 | ||||
Kd | 7.35 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.21 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.17 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.13 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.01 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 6.45 | J Med Chem, (2017) 60:9:4002 | ||||
TAF1
Transcription initiation factor TFIID subunit 1
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.89 | |||||
IC50 | 8.1 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.96 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.89 | J Med Chem, (2017) 60:1:157 | ||||
Kd | 7.78 | J Med Chem, (2017) 60:9:4002 | ||||
IC50 | 7.77 | J Med Chem, (2017) 60:9:4002 | ||||