Pharos : Ligand Details

Target Activities

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1 – 7 of 7

SIGMAR1

Tclin

Sigma non-opioid intracellular receptor 1

3 Activities

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1 – 3 of 3

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	7.54	None, None:None:None

Ki	7.92	None, None:None:None

Ki	8.1	J. Med. Chem., (2005) 48:15:4754	16033255

SLC6A2

Tclin

Sodium-dependent noradrenaline transporter

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Activity Reference
IC50	6.06	None, None:None:None

Ki	6.07	None, None:None:None

ESR1

Tclin

Estrogen receptor

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Activity Reference
IC50	8.34	None, None:None:None

Ki	8.88	None, None:None:None

SLC6A4

Tclin

Sodium-dependent serotonin transporter

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Activity Reference
IC50	6.2	None, None:None:None

Ki	6.47	None, None:None:None

SLC6A3

Tclin

Sodium-dependent dopamine transporter

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Activity Reference
IC50	6.11	None, None:None:None

Ki	6.21	None, None:None:None

PTGS1

Tclin

Prostaglandin G/H synthase 1

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.46		None, None:None:None

EBP

Tchem

3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	9		J. Med. Chem., (2005) 48:15:4754	16033255