Pharos : Ligand Details - JCJR52WLRN2J

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Ligand Summary

Ligand Structure

chemical structure image

Synonyms & Links

Name: Clomiphene

PubChem: 1548953

ChEMBL: CHEMBL954

LyCHI: JCJR52WLRN2J

Target Activities

SIGMAR1

Tclin

Sigma non-opioid intracellular receptor 1

3 Activities

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1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.54		None, None:None:None

Ki	7.92		None, None:None:None

Ki	8.1		J. Med. Chem., (2005) 48:15:4754	16033255

SLC6A2

Tclin

Sodium-dependent noradrenaline transporter

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.06		None, None:None:None

Ki	6.07		None, None:None:None

ESR1

Tclin

Estrogen receptor

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.34		None, None:None:None

Ki	8.88		None, None:None:None

SLC6A4

Tclin

Sodium-dependent serotonin transporter

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.2		None, None:None:None

Ki	6.47		None, None:None:None

SLC6A3

Tclin

Sodium-dependent dopamine transporter

2 Activities

Items per page:

1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.11		None, None:None:None

Ki	6.21		None, None:None:None

PTGS1

Tclin

Prostaglandin G/H synthase 1

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.46		None, None:None:None

EBP

Tchem

3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	9		J. Med. Chem., (2005) 48:15:4754	16033255