Clomiphene
Ligand Summary
Target Activities
SIGMAR1
Sigma non-opioid intracellular receptor 1
3 Activities
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1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.1 | J. Med. Chem., (2005) 48:15:4754 | ||||
Ki | 7.92 | None, None:None:None | ||||
IC50 | 7.54 | None, None:None:None | ||||
SLC6A4
Sodium-dependent serotonin transporter
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.47 | None, None:None:None | ||||
IC50 | 6.2 | None, None:None:None | ||||
SLC6A3
Sodium-dependent dopamine transporter
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.21 | None, None:None:None | ||||
IC50 | 6.11 | None, None:None:None | ||||
ESR1
Estrogen receptor
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.88 | None, None:None:None | ||||
IC50 | 8.34 | None, None:None:None | ||||
SLC6A2
Sodium-dependent noradrenaline transporter
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.07 | None, None:None:None | ||||
IC50 | 6.06 | None, None:None:None | ||||
PTGS1
Prostaglandin G/H synthase 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.46 | None, None:None:None | ||||
EBP
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9 | J. Med. Chem., (2005) 48:15:4754 | ||||