rocaglamide
Ligand Summary
Target Activities
RELA
Transcription factor p65
5 Activities
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1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.16 | Bioorg Med Chem, (2018) 26:15:4452 | ||||
IC50 | 7.12 | J. Nat. Prod., (2011) 74:5:1117 | ||||
IC50 | 7.12 | J. Nat. Prod., (2011) 74:5:1126 | ||||
IC50 | 7.1 | J. Nat. Prod., (2009) 72:11:2028 | ||||
IC50 | 6.92 | J Nat Prod, (2019) 82:6:1645 | ||||
EIF4A1
Eukaryotic initiation factor 4A-I
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 8.33 | J Med Chem, (2020) 63:11:5879 | ||||
IC50 | 7.33 | J Med Chem, (2020) 63:11:5879 | ||||
IC50 | 6.87 | J Med Chem, (2020) 63:11:5879 | ||||
Kd | 6.81 | J Med Chem, (2020) 63:11:5879 | ||||
IC50 | 6.64 | J Med Chem, (2020) 63:11:5879 | ||||
NFKB1
Nuclear factor NF-kappa-B p105 subunit
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.12 | J. Nat. Prod., (2010) 73:5:949 | ||||