US8877795, 12
Ligand Summary
Target Activities
PIM1
Serine/threonine-protein kinase pim-1
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.77 | J Med Chem, (2017) 60:7:2853 | ||||
IC50 | 7.62 | Bioorg. Med. Chem. Lett., (2009) 19:11:3019 | ||||
IC50 | 7.62 | J. Med. Chem., (2009) 52:1:74 | ||||
IC50 | 7.62 | J. Med. Chem., (2012) 55:6:2641 | ||||
Ki | 7.62 | J. Med. Chem., (2012) 55:19:8199 | ||||
TTR
Transthyretin
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.09 | None, (2014) None:None:None | ||||
CISD1
CDGSH iron-sulfur domain-containing protein 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.53 | Bioorg Med Chem Lett, (2016) 26:21:5350 | ||||