riviciclib
Ligand Summary
Name: riviciclib
PubChem: 23643976
PubChem: 23643975
Guide to Pharmacology: 7934
ChEMBL: CHEMBL3991935
LyCHI: HT2W9QA2CSJZ
Target Activities
CDK9
Cyclin-dependent kinase 9
2 Activities
CDK1
Cyclin-dependent kinase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.1 | |||||
CDK4
Cyclin-dependent kinase 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.2 | |||||
PLK1
Serine/threonine-protein kinase PLK1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.68 | Science, (2017) 358:6367:None | ||||
CDKL5
Cyclin-dependent kinase-like 5
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
DDX42
ATP-dependent RNA helicase DDX42
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.7 | Science, (2017) 358:6367:None | ||||