Linsitinib
Ligand Summary
Target Activities
IGF1R
Insulin-like growth factor 1 receptor
9 Activities
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1 – 9 of 9
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 8.7 | Eur. J. Med. Chem., (2015) 92:None:246 | ||||
IC50 | 8.55 | Bioorg. Med. Chem. Lett., (2016) 26:8:2057 | ||||
IC50 | 8.12 | Bioorg. Med. Chem. Lett., (2016) 26:8:2057 | ||||
IC50 | 7.92 | ACS Med. Chem. Lett., (2013) 4:7:627 | ||||
IC50 | 7.89 | ACS Med. Chem. Lett., (2013) 4:7:627 | ||||
IC50 | 7.85 | Bioorg. Med. Chem. Lett., (2016) 26:8:2057 | ||||
IC50 | 7.75 | Bioorg. Med. Chem. Lett., (2010) 20:8:2452 | ||||
IC50 | 7.62 | Bioorg. Med. Chem. Lett., (2011) 21:4:1176 | ||||
IC50 | 7.62 | ACS Med. Chem. Lett., (2013) 4:7:627 | ||||
INSR
Insulin receptor
2 Activities
MAPK11
Mitogen-activated protein kinase 11
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 8 | Science, (2017) 358:6367:None | ||||
ABCG2
ATP-binding cassette sub-family G member 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | 6.98 | Eur J Med Chem, (2019) 164:None:193 | ||||