danusertib
Ligand Summary
Name: danusertib
PubChem: 11442891
Guide to Pharmacology: 7937
ChEMBL: CHEMBL402548
LyCHI: HK1TZGJHTVSP
Target Activities
AURKA
Aurora kinase A
14 Activities
Items per page:
1 – 10 of 14
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.89 | |||||
Kd | 8.67 | None, None:None:None | ||||
Ki | 8.6 | J. Med. Chem., (2006) 49:24:7247 | ||||
Kd | 8.57 | None, None:None:None | ||||
Kd | 8.47 | None, None:None:None | ||||
Kd | 8.43 | None, None:None:None | ||||
Kd | 8.4 | None, None:None:None | ||||
Kd | 8.01 | None, None:None:None | ||||
Kd | 7.96 | Science, (2017) 358:6367:None | ||||
IC50 | 7.89 | J. Med. Chem., (2006) 49:24:7247 | ||||
ABL1
Tyrosine-protein kinase ABL1
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.3 | J. Med. Chem., (2010) 53:15:5439 | ||||
IC50 | 8.1 | J. Med. Chem., (2013) 56:17:6991 | ||||
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
IC50 | 7.6 | J. Med. Chem., (2006) 49:24:7247 | ||||
AURKB
Aurora kinase B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.1 | |||||
AURKC
Aurora kinase C
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.21 | |||||
SLK
STE20-like serine/threonine-protein kinase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.21 | |||||
PRKAG2
5'-AMP-activated protein kinase subunit gamma-2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.03 | Science, (2017) 358:6367:None | ||||
FYN
Tyrosine-protein kinase Fyn
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
EPHA2
Ephrin type-A receptor 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.62 | Science, (2017) 358:6367:None | ||||
ABL2
Tyrosine-protein kinase ABL2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8 | Science, (2017) 358:6367:None | ||||
BCR
Breakpoint cluster region protein
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
NUAK2
NUAK family SNF1-like kinase 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.6 | Science, (2017) 358:6367:None | ||||
ERCC2
General transcription and DNA repair factor IIH helicase subunit XPD
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.87 | Science, (2017) 358:6367:None | ||||
RET
Proto-oncogene tyrosine-protein kinase receptor Ret
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.22 | Science, (2017) 358:6367:None | ||||
PLK4
Serine/threonine-protein kinase PLK4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.3 | Science, (2017) 358:6367:None | ||||
EPHB4
Ephrin type-B receptor 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.75 | Science, (2017) 358:6367:None | ||||