Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzyl)amide Bis-(trifluoroacetate)
Ligand Summary
Name: Benzylsulfonyl-D-argininyl-proline-(4-amidinobenzyl)amide Bis-(trifluoroacetate)
PubChem: 46899577
PubChem: 49864062
Guide to Pharmacology: 8670
ChEMBL: CHEMBL1215083
ChEMBL: CHEMBL1229259
LyCHI: HACKCQ3JCNAV
Target Activities
TMPRSS6
Transmembrane protease serine 6
3 Activities
TMPRSS11D
Transmembrane protease serine 11D
2 Activities
TMPRSS2
Transmembrane protease serine 2
2 Activities
F2
Prothrombin
2 Activities
ST14
Suppressor of tumorigenicity 14 protein
2 Activities
PLG
Plasminogen
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.41 | Bioorg. Med. Chem. Lett., (2011) 21:16:4860 | ||||
KLKB1
Plasma kallikrein
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.08 | Bioorg. Med. Chem. Lett., (2011) 21:16:4860 | ||||
F10
Coagulation factor X
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.62 | Bioorg. Med. Chem. Lett., (2011) 21:16:4860 | ||||