Pharos : Ligand Details - H9SSQYFZL1HD

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: combretastatin A4

PubChem: 5351344

Guide to Pharmacology: 8854

ChEMBL: CHEMBL67

LyCHI: H9SSQYFZL1HD

Target Activities

Explore Associated and Predicted Targets

TUBB3

Tclin

Tubulin beta-3 chain

3 Activities

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1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.24			23895532

IC50	8.28		Bioorg. Med. Chem., (2013) 21:4:891	23332369

IC50	8.24		J. Med. Chem., (2013) 56:17:6829	23895532

ABCB1

Tchem

Multidrug resistance protein 1

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.18		J. Med. Chem., (2013) 56:17:6829	23895532

IC50	7.94		Bioorg. Med. Chem., (2013) 21:4:891	23332369

TUBB1

Tclin

Tubulin beta-1 chain

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.75		J. Med. Chem., (2005) 48:2:457	15658859