BMS-681
Ligand Summary
Name: BMS-681
PubChem: 68764898
Guide to Pharmacology: 9430
ChEMBL: CHEMBL3577945
LyCHI: H7Z8P1BNXHNT
Target Activities
CCR2
C-C chemokine receptor type 2
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9.15 | |||||
IC50 | 9.62 | ACS Med. Chem. Lett., (2015) 6:4:439 | ||||
IC50 | 9.15 | ACS Med. Chem. Lett., (2015) 6:4:439 | ||||
IC50 | 9.15 | ACS Med Chem Lett, (2019) 10:3:300 | ||||
IC50 | 8.33 | ACS Med. Chem. Lett., (2015) 6:4:439 | ||||
CCR5
C-C chemokine receptor type 5
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.62 | |||||
IC50 | 8.62 | ACS Med. Chem. Lett., (2015) 6:4:439 | ||||
IC50 | 8.62 | ACS Med Chem Lett, (2019) 10:3:300 | ||||
IC50 | 8.37 | ACS Med. Chem. Lett., (2015) 6:4:439 | ||||
KCNH2
Potassium voltage-gated channel subfamily H member 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5.75 | ACS Med. Chem. Lett., (2015) 6:4:439 | ||||