Pharos : Ligand Details - H7Z8P1BNXHNT

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: BMS-681

PubChem: 68764898

Guide to Pharmacology: 9430

ChEMBL: CHEMBL3577945

LyCHI: H7Z8P1BNXHNT

Target Activities

Explore Associated and Predicted Targets

CCR2

Tchem

C-C chemokine receptor type 2

5 Activities

Items per page:

1 – 5 of 5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	9.15			25893046

IC50	9.62		ACS Med. Chem. Lett., (2015) 6:4:439	25893046

IC50	9.15		ACS Med. Chem. Lett., (2015) 6:4:439	25893046

IC50	9.15		ACS Med Chem Lett, (2019) 10:3:300	30891130

IC50	8.33		ACS Med. Chem. Lett., (2015) 6:4:439	25893046

CCR5

Tclin

C-C chemokine receptor type 5

4 Activities

Items per page:

1 – 4 of 4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.62			25893046

IC50	8.62		ACS Med. Chem. Lett., (2015) 6:4:439	25893046

IC50	8.62		ACS Med Chem Lett, (2019) 10:3:300	30891130

IC50	8.37		ACS Med. Chem. Lett., (2015) 6:4:439	25893046

KCNH2

Tclin

Potassium voltage-gated channel subfamily H member 2

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	5.75		ACS Med. Chem. Lett., (2015) 6:4:439	25893046