CHEMBL3289410
Ligand Summary
Name: N-[3-(Dimethylamino)propyl]-12-oxo-12H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxamide
PubChem: 90644346
ChEMBL: CHEMBL3289410
LyCHI: H6T12PFFAD8G
Target Activities
POLR1A
DNA-directed RNA polymerase I subunit RPA1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.37 | J. Med. Chem., (2014) 57:11:4950 | ||||