CHEMBL248176
Ligand Summary
NCATS Inxight: Drugs: 16129582
Name: 4-(5-chloro-4-(1H-indol-3-yl)pyrimidin-2-ylamino)-N-ethylpiperidine-1-carboxamide
PubChem: 16129582
ChEMBL: CHEMBL248176
LyCHI: GRCSHC1HY44J
Target Activities
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JUN
Transcription factor AP-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.15 | Bioorg. Med. Chem. Lett., (2007) 17:12:3463 | ||||
MAPK9
Mitogen-activated protein kinase 9
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.6 | Bioorg. Med. Chem. Lett., (2007) 17:12:3463 | ||||
MAPK8
Mitogen-activated protein kinase 8
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.89 | Bioorg. Med. Chem. Lett., (2007) 17:12:3463 | ||||