Pharos : Ligand Details - GQ1R63CA6PK3

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: CHEMBL4588728

PubChem: 155567528

ChEMBL: CHEMBL4588728

LyCHI: GQ1R63CA6PK3

Target Activities

Explore Associated and Predicted Targets

SCN1A

Tclin

Sodium channel protein type 1 subunit alpha

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	7.43		J Med Chem, (2019) 62:19:8695	31012583

SCN5A

Tclin

Sodium channel protein type 5 subunit alpha

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.1		J Med Chem, (2019) 62:19:8695	31012583

SCN4A

Tclin

Sodium channel protein type 4 subunit alpha

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.85		J Med Chem, (2019) 62:19:8695	31012583

SCN2A

Tclin

Sodium channel protein type 2 subunit alpha

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.92		J Med Chem, (2019) 62:19:8695	31012583

SCN8A

Tclin

Sodium channel protein type 8 subunit alpha

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.89		J Med Chem, (2019) 62:19:8695	31012583

SCN3A

Tclin

Sodium channel protein type 3 subunit alpha

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	6.68		J Med Chem, (2019) 62:19:8695	31012583

SCN7A

Tclin

Sodium channel protein type 7 subunit alpha

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	9.05		J Med Chem, (2019) 62:19:8695	31012583